MPEP

目录号: A12589

mGlu5 receptor antagonist

MPEP Chemical Structure

CAS NO. 96206-92-7

MPEP is a potent and highly selective non-competitive antagonist at the mGlu5 receptor subtype (IC50 = 36 nM) and a positive allosteric modulator at mGlu4 receptors.

库存: 现货

规格 价格 数量
10 mg
¥ 500.00
25 mg
¥ 1,000.00
50 mg
¥ 1,600.00
100 mg
¥ 2,800.00
10mM * 1mL in DMSO
¥ 700.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

MPEP is a potent and highly selective non-competitive antagonist at the mGlu5 receptor subtype (IC50 = 36 nM) and a positive allosteric modulator at mGlu4 receptors.
Targets
mGluR5
36 nM
In vitro DMSO 39 mg/mL (201.82 mM)
Water <1 mg/mL (<1 mM)
Ethanol 39 mg/mL (201.82 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 51.75 mL 258.73 mL 517.47 mL
0.5 mM 10.35 mL 51.75 mL 103.49 mL
1 mM 5.17 mL 25.87 mL 51.75 mL
5 mM 1.03 mL 5.17 mL 10.35 mL

*The above data is based on the productmolecular weight 193.249. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A12589
MECHANISM OF ACTION Antagonist
M. Wt 193.249
Formula C14H11N
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 96206-92-7
Synonyms N/A
SMILES CC1=CC=CC(=N1)C#CC2=CC=CC=C2

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