Imofinostat (MPT0E028)
目录号: A18982
HDAC 抑制剂
MPT0E028 是一种口服活性且选择性的 HDAC 抑制剂,其 IC50 分别针对 HDAC1、HDAC2 和 HDAC6 为 53.0 nM、106.2 nM 和 29.5 nM。
Discription | MPT0E028 is an orally active and selective HDAC inhibitor with IC50s of 53.0 nM, 106.2 nM, 29.5 nM for HDAC1, HDAC2 and HDAC6, respectively. | ||
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目录号 | A18982 |
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分子式 | C17H16N2O4S |
分子量 | 344.38 |
CAS号 | 1338320-94-7 |
SMILES | O=C(/C=C/C1=CC2=C(C=C1)N(CC2)S(=O)(C3=CC=CC=C3)=O)NO |
其他名称 | MPT-0E028 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2