MT-3014
目录号: A18580
PDE 10A 抑制剂
MT-3014 是一种强效、高选择性且能穿透大脑的磷酸二酯酶 10A(PDE 10A)抑制剂,其对人类 PDE 10A 和牛 PDE 10A 的 IC50 分别为 0.062 nM 和 0.09 nM。
Discription | MT-3014 is a potent, highly selective and brain-penetrated phosphodiesterase 10A (PDE 10A) inhibitor, with IC50s of 0.062 nM and 0.09 nM for human PDE 10A and bovine PDE 10A, respectively. | ||
---|---|---|---|
Targets |
|
目录号 | A18580 |
---|---|
分子式 | C23H25F2N7O |
分子量 | 453.49 |
CAS号 | 1332727-40-8 |
SMILES | CC(O)(C)CNC1=CC(N2C[C@H](F)CC2)=NC3=CC(C4=NC5=CC(F)=CC=C5N=C4C)=NN13 |
其他名称 | MT3014, MT 3014 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2