MT-802
目录号: A18589
BTK degrader
MT-802 是一种基于 PROTAC 技术的强效 BTK 降解剂,其 DC50 为 1 nM。MT-802 有潜力治疗 C481S 突变型慢性淋巴细胞白血病(CLL)。
Discription | MT-802 is a potent BTK degrader based on PROTAC technology, with a DC50 of 1 nM. MT-802 has potential to treat C481S mutant chronic lymphocytic leukemia (CLL). |
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目录号 | A18589 |
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分子式 | C41H41N9O8 |
分子量 | 787.82 |
CAS号 | 2231744-29-7 |
SMILES | O=C(NC1=CC2=C(C(N(C(CC3)C(NC3=O)=O)C2=O)=O)C=C1)COCCOCCN4CCC(N5N=C(C6=CC=C(OC7=CC=CC=C7)C=C6)C8=C(N)N=CN=C85)CC4 |
其他名称 | MT802, MT 802 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2