Mutant IDH1-IN-2
目录号: A21339
IDH 抑制剂
Mutant IDH1-IN-2 是一种突变型异柠檬酸脱氢酶(IDH)蛋白的抑制剂,在LS-MS生化测定中具有IC50,在荧光生化测定中的IC50为16.6 nM。
| Discription | Mutant IDH1-IN-2 is a inhibitor of mutant Isocitrate dehydrogenase (IDH) proteins, with IC50 of in LS-MS biochemical assay, IC50 of 16.6 nM in Fluorescence biochemical assay. |
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| 目录号 | A21339 |
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| 分子式 | C24H31F2N5O2 |
| 分子量 | 459.53 |
| CAS号 | 1429176-69-1 |
| SMILES | O=C1OC[C@H](C(C)C)N1C2=NC(N[C@H](C3=CC=C(CN4CCC(F)(F)CC4)C=C3)C)=NC=C2 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2