Nelotanserin
目录号: A21506
5-HT2A inverse 激动剂
Nelotanserin 是一种强效的 5-HT2A 反向激动剂,中等强度的 5-HT2C 部分反向激动剂,以及弱效的 5-HT2B 反向激动剂,在 IP 积累实验中,其 IC50 分别为 1.7、79、791 纳摩尔。
Discription | Nelotanserin is a potent 5-HT2A inverse agonist, a moderately potent 5-HT2C partial inverse agonist and a weak 5-HT2B inverse agonist, with IC50s of 1.7, 79, 791 nM in IP accumulation assays, respectively. | ||
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目录号 | A21506 |
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分子式 | C18H15BrF2N4O2 |
分子量 | 437.24 |
CAS号 | 839713-36-9 |
SMILES | COC1=C(C2=C(Br)C=NN2C)C=C(NC(NC3=C(F)C=C(F)C=C3)=O)C=C1 |
其他名称 | APD125, APD 125, APD-125 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2