Netupitant

目录号: A14428

NK1 receptor antagonist

Netupitant Chemical Structure

CAS NO. 290297-26-6

Netupitant is a selective neurokinin 1 (NK1) receptor antagonist. It competitively binds to and blocks the activity of the human substance P/NK1 receptors in the central nervous system (CNS), thereby inhibiting NK1-receptor binding of the endogenous tachykinin neuropeptide substance P (SP), which may result in the prevention of chemotherapy-induced nausea and vomiting (CINV).

库存: 现货

规格 价格 数量
5 mg
¥ 400.00
10 mg
¥ 700.00
25 mg
¥ 1,500.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

Netupitant is a selective neurokinin 1 (NK1) receptor antagonist. It competitively binds to and blocks the activity of the human substance P/NK1 receptors in the central nervous system (CNS), thereby inhibiting NK1-receptor binding of the endogenous tachykinin neuropeptide substance P (SP), which may result in the prevention of chemotherapy-induced nausea and vomiting (CINV).
Targets
neurokinin 1 receptor
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.28 mL 86.42 mL 172.83 mL
0.5 mM 3.46 mL 17.28 mL 34.57 mL
1 mM 1.73 mL 8.64 mL 17.28 mL
5 mM 0.35 mL 1.73 mL 3.46 mL

*The above data is based on the productmolecular weight 578.59. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A14428
MECHANISM OF ACTION Antagonist
M. Wt 578.59
Formula C30H32F6N4O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 290297-26-6
Synonyms D05152, AG-E-94200
SMILES CC1=CC=CC=C1C2=CC(=NC=C2N(C)C(=O)C(C)(C)C3=CC(=CC(=C3)C(F)(F)F)C(F)(F)F)N4CCN(CC4)C

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