NVP-BAG956
目录号: A11511
PI3K/PDK-1 抑制剂
NVP-BAG956 作为一种强效、可逆的、与ATP竞争的 PI 3-K/PDK1 双激酶抑制剂,对 VEGFR1 的抑制效力较低(IC50 = 2.56 uM),对其他15种激酶的活性几乎没有或完全没有(IC50 >10 uM)。
Discription | NVP-BAG956 acts as a potent, reversible, and ATP-competitive PI 3-K/PDK1 dual kinase inhibitor, displaying much reduced potency against VEGFR1 (IC50 = 2.56 uM) and little or no activity toward a panel of 15 other kinases (IC50 >10 uM). | ||
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目录号 | A11511 |
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分子式 | C28H21N5 |
分子量 | 427.5 |
CAS号 | 853910-02-8 |
SMILES | CC1=NC2=CN=C3C=CC(=CC3=C2N1C4=CC=C(C=C4)C(C)(C)C#N)C#CC5=CN=CC=C5 |
其他名称 | NVP-BAG 956 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2