Olcegepant
目录号: A11512
CGRP1 receptor
Olcegepant 是一种强效且选择性的非肽类拮抗剂,针对 钙调素基因相关肽1 (CGRP1) 受体,具有 0.03 nM 的 IC50 和针对人类 CGRP 的 14.4 pM 的 Ki。
Discription | Olcegepant is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP. | |||||
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Cell Research |
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目录号 | A11512 |
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分子式 | C38H47Br2N9O5 |
分子量 | 869.65 |
CAS号 | 204697-65-4 |
SMILES | O=C1N(CC2=C(N1)C=CC=C2)C3CCN(C(N[C@@H](C(N[C@H](C(N4CCN(C5=CC=NC=C5)CC4)=O)CCCCN)=O)CC6=CC(Br)=C(C(Br)=C6)O)=O)CC3 |
其他名称 | BIBN-4096; BIBN 4096BS |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2