OTX015

目录号: A13890

BET inhibitor

OTX015

OTX015 Chemical Structure

CAS NO. 202590-98-5

OTX015 is an orally bioavailable, small molecule inhibitor of BRD2, BRD3, and BRD4 (EC50s = 10-19 nM).

库存: 现货

规格 价格 数量
5 mg
¥ 700.00
10 mg
¥ 900.00
25 mg
¥ 1,800.00
50 mg
¥ 2,500.00
10mM * 1mL in DMSO
¥ 1,300.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

OTX015 is an orally bioavailable, small molecule inhibitor of BRD2, BRD3, and BRD4 (EC50s = 10-19 nM).
Targets
BRDs (Cell-free assay)
10-19 nM(EC50)
In vitro DMSO 98 mg/mL (199.19 mM)
Water <1 mg/mL (<1 mM)
Ethanol 98 mg/mL (199.19 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.33 mL 101.63 mL 203.26 mL
0.5 mM 4.07 mL 20.33 mL 40.65 mL
1 mM 2.03 mL 10.16 mL 20.33 mL
5 mM 0.41 mL 2.03 mL 4.07 mL

*The above data is based on the productmolecular weight 491.99. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Technical Details

目录号 A13890
MECHANISM OF ACTION Inhibitor
M. Wt 491.99
Formula C25H22ClN5O2S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 202590-98-5
Synonyms OTX 015, OTX-015
SMILES CC1=C(SC2=C1C(=N[C@H](C3=NN=C(N32)C)CC(=O)NC4=CC=C(C=C4)O)C5=CC=C(C=C5)Cl)C

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