Parsaclisib

Name: Parsaclisib
SKU: A13561

目录号: A13561

PI3Kδ inhibitor

Parsaclisib Chemical Structure

CAS NO. 1426698-88-5

Parsaclisib is a potent and selective PI3Kδ inhibitor, with an IC50 of 1 nM at 1 mM ATP, and shows appr 20,000-fold selectivity for PI3Kα, PI3Kβ, PI3Kγ and 57 other kinases.

库存：现货

规格	价格	数量
5 mg	￥ 4,500.00
10 mg	￥ 7,750.00
50 mg	￥ 23,000.00
100 mg	￥ 46,000.00

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生物活性

Parsaclisib is a potent and selective PI3Kδ inhibitor, with an IC50 of 1 nM at 1 mM ATP, and shows appr 20,000-fold selectivity for PI3Kα, PI3Kβ, PI3Kγ and 57 other kinases.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	23.1 mL	115.51 mL	231.01 mL
0.5 mM	4.62 mL	23.1 mL	46.2 mL
1 mM	2.31 mL	11.55 mL	23.1 mL
5 mM	0.46 mL	2.31 mL	4.62 mL

*The above data is based on the productmolecular weight 432.88. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A13561
作用机制	Inhibitor (抑制剂)
M. Wt	432.88
Formula	C20H22ClFN6O2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1426698-88-5
Synonyms	INCB050465, INCB-050465, INCB 050465
SMILES	CCOC1=C([C@@H](C2)CNC2=O)C(F)=C(Cl)C=C1[C@@H](N3C4=NC=NC(N)=C4C(C)=N3)C