PD 123319 ditrifluoroacetate

Name: PD 123319 ditrifluoroacetate
SKU: A13201
Price: 420 CNY
Rating: 5 (1 reviews)

目录号: A13201

angiotensin AT2 receptor 拮抗剂

1 篇发表文献

PD 123319 ditrifluoroacetate 是一种强效的、选择性的、非肽类血管紧张素 AT2 受体拮抗剂。在大鼠肾上腺组织和大脑中的 IC50 值分别为 34 nM 和 210 nM。

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Grouped product items
规格	价格	库存
5mg	¥420.00	现货
10mg	¥805.00	现货
25mg	¥1,645.00	现货
50mg	¥2,765.00	现货
100mg	¥4,865.00	现货
200mg	¥6,930.00	现货
*10mM 1mL in DMSO**	¥980.00	现货
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Data Sheet

SDS

顾客使用 Adooq 产品发表的高质量科研文献

Adooq用户使用PD 123319 ditrifluoroacetate发表的1篇文献

Dao-Lai Zhang, .et al. , eLife, 2018, 7: e33432 PMID: 29393851

生物活性

Discription

PD 123319 ditrifluoroacetate is a potent, selective, non-peptide angiotensin AT2 receptor antagonist. IC50 values are 34 and 210 nM in rat adrenal tissue and brain respectively.

Targets

Target	Value

产品信息

目录号	A13201
分子式	C31H32N4O3.2CF3CO2H
分子量	736.67
CAS号	136676-91-0 (TFA), 130663-39-7
SMILES	CC1=C(C=CC(=C1)CN2C=NC3=C2CC(N(C3)C(=O)C(C4=CC=CC=C4)C5=CC=CC=C5)C(=O)O)N(C)C.C(=O)(C(F)(F)F)O.C(=O)(C(F)(F)F)O
其他名称	PD123319, PD-123319
储存条件	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

溶解性数据

In vitro (25°C)	DMSO	87 mg/mL (171.05 mM)
	Water	87 mg/mL (171.05 mM)
	Ethanol	87 mg/mL (171.05 mM)
In vivo	Saline	28 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	13.57 mL	67.87 mL	135.75 mL
0.5 mM	2.71 mL	13.57 mL	27.15 mL
1 mM	1.36 mL	6.79 mL	13.57 mL
5 mM	0.27 mL	1.36 mL	2.71 mL

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