PD 151746

目录号: A14245

Calpain inhibitor

PD 151746 Chemical Structure

CAS NO. 179461-52-0

PD 151746 is a selective, cell-permeable calpain inhibitor with Ki of 0.26 uM for μ-Calpain, about 20-fold selectivity over m-calpain.

库存: 现货

规格 价格 数量
10 mg
¥ 900.00
25 mg
¥ 1,800.00
50 mg
¥ 3,000.00
10mM * 1mL in DMSO
¥ 950.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

PD 151746 is a selective, cell-permeable calpain inhibitor with Ki of 0.26 uM for μ-Calpain, about 20-fold selectivity over m-calpain.
Targets
μ-Calpain m-calpain
260 nM5.33 μM
In vitro DMSO 47 mg/mL (198.1 mM)
Water <1 mg/mL (<1 mM)
Ethanol 47 mg/mL (198.1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 42.15 mL 210.75 mL 421.5 mL
0.5 mM 8.43 mL 42.15 mL 84.3 mL
1 mM 4.21 mL 21.07 mL 42.15 mL
5 mM 0.84 mL 4.21 mL 8.43 mL

*The above data is based on the productmolecular weight 237.25. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A14245
MECHANISM OF ACTION Inhibitor
M. Wt 237.25
Formula C11H8FNO2S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 179461-52-0
Synonyms PD-151746,PD151746
SMILES C1=CC2=C(C=C1F)C(=CN2)/C=C(/C(=O)O)\S

产品标签

产品标签

其他人对该产品使用了下列标签:

使用空格分隔标签。使用单引号(')标注词组。

Product Questions

Product Questions

No Questions
Keywords:购买 PD 151746 | PD 151746 供应商 | 订购 PD 151746 | PD 151746 价格 | PD 151746 生产商 | 订单 PD 151746 | PD 151746 代理商 | 购买 179461-52-0| 179461-52-0 供应商 | 订购 179461-52-0 | 179461-52-0 价格 | 179461-52-0 生产商 | 订单 179461-52-0 | 179461-52-0 代理商|buy PD 151746 | PD 151746 Supplier | purchase PD 151746 | PD 151746 cost | PD 151746 manufacturer | order PD 151746 | PD 151746 distributor | buy 179461-52-0| 179461-52-0 Supplier | purchase 179461-52-0 | 179461-52-0 cost | 179461-52-0 manufacturer | order 179461-52-0 | 179461-52-0 distributor
Rewards