PDK1 inhibitor
目录号: A16185
PDK1 抑制剂
PDK1 抑制剂,强效、ATP 竞争性并且选择性的双 PI3K 和 PDPK1 抑制剂(IC50 值分别为 PDK1 和 p-T308-PKB 抑制为 34 nM 和 94 nM)。
Discription | PDK1 inhibitor, potent, ATP-competitive and selective dual PI3K and PDPK1 inhibitor (IC50 values 34 nM and 94 nM for PDK1 and p-T308-PKB inhibition, respectively. |
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目录号 | A16185 |
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分子式 | C25H15N5.HCl |
分子量 | 421.88 |
CAS号 | 853909-77-0 |
SMILES | C1=CC(=CN=C1)C#CC2=CC3=C4C(=CN=C3C=C2)N=CN4C5=CC=C(C=C5)CC#N.Cl |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2