PDK1

Catalog No.Inhibitor Name PDK-1 Other Targets
A10681OSU-03012
**
A11148BX-795
****
TBK1/IKKɛ,c-Kit,CDK2/CyclinE
A11149BX-912
***
PKA,KDR,CDK2/CyclinE
A11032PHT-427
*
Akt
A12767GSK2334470
***
A12881 BX-517
****
A11511NVP-BAG956
*
PI3K
A13484PS 48
*

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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  1. PS 48

    Catalog No. A13484
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    PDK1 抑制剂
    PS 48是一种变构磷酸肌醇依赖性蛋白激酶-1(PDK1)激活剂(Kd = 10.3μM)。 了解更多
  2. TEPP-46

    Catalog No. A16279
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    PKM2 activator
    TEPP-46是重组丙酮酸激酶M2(PKM2)的有效选择性活化剂,最大活化浓度(AC50值)的一半为92 nM,相对于PKM1,PKL和PKR几乎没有或没有活性。 了解更多

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