PF-04957325
目录号: A21246
PDE8 抑制剂
PF-04957325 是一种高效且选择性的 PDE8 抑制剂,其 IC50 分别为 PDE8A 的 0.7 nM 和 PDE8B 的 0.3 nM。
Discription | PF-04957325 is a highly potent and selective PDE8 inhibitor, with IC50s of 0.7 nM and 0.3 nM for PDE8A and PDE8B, respectively. |
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目录号 | A21246 |
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分子式 | C14H15F3N8OS |
分子量 | 400.38 |
CAS号 | 1305115-80-3 |
SMILES | NC1=C(N=NN2C[C@H]3CN(CC4=NC=CS4)CCO3)C2=NC(C(F)(F)F)=N1 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2