PF-06250112
目录号: A18612
BTK 抑制剂
PF-06250112 是一种高效、高选择性、口服生物利用度的 BTK 抑制剂,其 IC50 为 0.5 nM,对 BMX 非受体酪氨酸激酶和 TEC 显示出抑制效果,其 IC50 分别为 0.9 nM 和 1.2 nM。
Discription | PF-06250112 is a potent, highly selective, orally bioavailable BTK inhibitor with an IC50 of 0.5 nM, shows inhibitory effect toward BMX nonreceptor tyrosine kinase and TEC with IC50s of 0.9 nM and 1.2 nM, respectively. |
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目录号 | A18612 |
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分子式 | C22H20F2N6O2 |
分子量 | 438.43 |
CAS号 | 1609465-89-5 |
SMILES | O=C(N)C1=C(N(N=C1C2=CC=C(C=C2)OC3=CC=C(C=C3F)F)[C@@H]4CN(CCC4)C#N)N |
其他名称 | PF06250112, PF 06250112 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2