PF-06273340
目录号: A22377
pan-Trk 抑制剂
PF-06273340 是一种高效、选择性强、耐受性好的全面 Trk 抑制剂,其 IC50 值分别针对 TrkA、TrkB、TrkC 为 6、4、3 nM。
Discription | PF-06273340 is a highly potent, kinases elective, well-tolerated pan-Trk inhibitor with IC50 values of 6, 4, 3 nM for TrkA, TrkB, Trk C, respectively. |
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目录号 | A22377 |
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分子式 | C23H22ClN7O3 |
分子量 | 479.92 |
CAS号 | 1402438-74-7 |
SMILES | CC(C)(CO)N1C=C(C2=CN=C(N=C21)N)C(=O)C3=CC(=CN=C3)NC(=O)CC4=NC=C(C=C4)Cl |
其他名称 | PF06273340,PF 06273340 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2