PF-06751979
目录号: A20066
BACE1 抑制剂
PF-06751979 是一种强效的、能穿透大脑的 β-位点淀粉前体蛋白裂解酶1 (BACE1) 抑制剂,在 BACE1 结合实验中的 IC50 为 7.3 nM。
Discription | PF-06751979 is a potent, brain penetrant, β-site amyloid precursor protein cleaving enzyme 1 (BACE1) inhibitor with an IC50 of 7.3 nM in BACE1 binding assay. | |||||
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Cell Research |
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目录号 | A20066 |
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分子式 | C18H19F2N5O3S2 |
分子量 | 455.5 |
CAS号 | 1818339-66-0 |
SMILES | FC(F)OC1=CN=C(C(NC2=CSC([C@]34CO[C@@H](C)C[C@@]3([H])CSC(N)=N4)=N2)=O)C=C1 |
其他名称 | PF 06751979, PF06751979 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2