PF-4

目录号: A13451

BRPF1 bromodomain inhibitor

PF-4 Chemical Structure

CAS NO. 900305-37-5

PFI-4 is a potent and selective and cell permeable BRPF1 bromodomain inhibitor (IC50 = 80 nM). Exhibits >100-fold selectivity for BRPF1 over a panel of other bromodomains including BRPF2 (BRD1), BRPF3 and BRD4.

库存: 现货

规格 价格 数量
10 mg
¥ 900.00
25 mg
¥ 1,900.00
50 mg
¥ 3,400.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

PFI-4 is a potent and selective and cell permeable BRPF1 bromodomain inhibitor (IC50 = 80 nM). Exhibits >100-fold selectivity for BRPF1 over a panel of other bromodomains including BRPF2 (BRD1), BRPF3 and BRD4.
Targets
BRPF1 BRPF2 BRPF3
80 nM7.9 μM>10μM
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 26.29 mL 131.43 mL 262.85 mL
0.5 mM 5.26 mL 26.29 mL 52.57 mL
1 mM 2.63 mL 13.14 mL 26.29 mL
5 mM 0.53 mL 2.63 mL 5.26 mL

*The above data is based on the productmolecular weight 380.44. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A13451
MECHANISM OF ACTION
M. Wt 380.44
Formula C21H24N4O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 900305-37-5
Synonyms PF4, PF 4
SMILES [H]N(C(C1=CC=CC=C1OC)=O)C2=C(N3CCCC3)C=C(N(C)C(N4C)=O)C4=C2

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