PF-AKT400
目录号: A21991
Akt 抑制剂
PF-AKT400 是一种广泛选择性、高效、与ATP竞争的Akt抑制剂,对PKBα(IC50=0.5 nM)的选择性比对PKA(IC50=450 nM)高出900倍。
Discription | PF-AKT400 is a broadly selective, potent, ATP-competitive Akt inhibitor, displays 900-fold greater selectivity for PKBα (IC50=0.5 nM) than PKA (IC50=450 nM). | |||||
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Cell Research |
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目录号 | A21991 |
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分子式 | C20H22F2N6O |
分子量 | 400.43 |
CAS号 | 1004990-28-6 |
SMILES | N[C@@](CC1)(CNC(C2=CC=C(F)C=C2F)=O)CN1C3=C4C(NC=C4CC)=NC=N3 |
其他名称 | AKT protein kinase inhibitor; PF-AKT400; PFAKT400; Lig1; Lig-1; Lig 1; PF AKT400; AKT-0286; AKT 0286; AKT0286 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2