PFI-2
目录号: A14216
SETD7 抑制剂
PFI-2 是一种强效、选择性且在细胞内活跃的赖氨酸甲基转移酶SETD7抑制剂,其Ki (app) 和 IC50 分别为0.33 nM 和 2 nM,对其他甲基转移酶和非表观遗传靶标具有1000倍的选择性。
Discription | PFI-2 is a potent, selective, and cell-active lysine methyltransferase SETD7 inhibitor with Ki (app) and IC50 of 0.33 nM and 2 nM, 1000-fold selectivity over other methyltransferases and other non-epigenetic targets. | ||
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目录号 | A14216 |
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分子式 | C23H25F4N3O3S |
分子量 | 499.52 |
CAS号 | 1627676-59-8 |
SMILES | C1CCN(C1)C(=O)[C@@H](CC2=CC(=CC=C2)C(F)(F)F)NS(=O)(=O)C3=CC(=C4CNCCC4=C3)F |
其他名称 | PFI2 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2