PFI-2

目录号: A14216

SETD7 抑制剂

PFI-2 Chemical Structure

CAS NO. 1627676-59-8

PFI-2 is a potent, selective, and cell-active lysine methyltransferase SETD7 inhibitor with Ki (app) and IC50 of 0.33 nM and 2 nM, 1000-fold selectivity over other methyltransferases and other non-epigenetic targets.

库存: 现货

规格 价格 数量
10 mg
¥ 1,000.00
25 mg
¥ 2,000.00
50 mg
¥ 3,500.00
10mM * 1mL in DMSO
¥ 1,050.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

PFI-2 is a potent, selective, and cell-active lysine methyltransferase SETD7 inhibitor with Ki (app) and IC50 of 0.33 nM and 2 nM, 1000-fold selectivity over other methyltransferases and other non-epigenetic targets.
靶点信息
SETD7 SETD7
0.33 nM(Ki)2 nM
In vitro DMSO 99 mg/mL (198.19 mM)
Water 4 mg/mL heating (8.0 mM)
Ethanol 66 mg/mL heating (132.12 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.02 mL 100.1 mL 200.19 mL
0.5 mM 4 mL 20.02 mL 40.04 mL
1 mM 2 mL 10.01 mL 20.02 mL
5 mM 0.4 mL 2 mL 4 mL

*The above data is based on the productmolecular weight 499.52. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A14216
MECHANISM OF ACTION Inhibitor
M. Wt 499.52
Formula C23H25F4N3O3S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1627676-59-8
Synonyms PFI2
SMILES C1CCN(C1)C(=O)[C@@H](CC2=CC(=CC=C2)C(F)(F)F)NS(=O)(=O)C3=CC(=C4CNCCC4=C3)F

产品标签

产品标签

其他人对该产品使用了下列标签:

使用空格分隔标签。使用单引号(')标注词组。

Product Questions

Product Questions

No Questions
Keywords:购买 PFI-2 | PFI-2 供应商 | 订购 PFI-2 | PFI-2 价格 | PFI-2 生产商 | 订单 PFI-2 | PFI-2 代理商 | 购买 1627676-59-8| 1627676-59-8 供应商 | 订购 1627676-59-8 | 1627676-59-8 价格 | 1627676-59-8 生产商 | 订单 1627676-59-8 | 1627676-59-8 代理商|buy PFI-2 | PFI-2 Supplier | purchase PFI-2 | PFI-2 cost | PFI-2 manufacturer | order PFI-2 | PFI-2 distributor | buy 1627676-59-8| 1627676-59-8 Supplier | purchase 1627676-59-8 | 1627676-59-8 cost | 1627676-59-8 manufacturer | order 1627676-59-8 | 1627676-59-8 distributor
Rewards