PFK15
目录号: A14287
PFKFB3 抑制剂
PFK15 是一种强效且选择性的 6-磷酸果糖-2-激酶(PFKFB3)抑制剂,其半抑制浓度(IC50)为207纳摩尔。
| Discription | PFK15 is a potent and selective 6-phosphofructo-2-kinase (PFKFB3) with IC50 of 207 nM. | ||
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| 目录号 | A14287 |
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| 分子式 | C17H12N2O |
| 分子量 | 260.29 |
| CAS号 | 4382-63-2 |
| SMILES | C1=CC=C2C(=C1)C=CC(=N2)/C=C/C(=O)C3=CC=NC=C3 |
| 其他名称 | PFK-015 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
| In vitro (25°C) | DMSO | Warmed: 17 mg/mL (65.31 mM) | |
| Water | Insoluble | ||
| Ethanol | Warmed: 2 mg/mL | ||
| In vivo | 5% DMSO+40% PEG 300+5% Tween 80+50% ddH2O | 2 mg/mL | |
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 38.42 mL | 192.09 mL | 384.19 mL |
| 0.5 mM | 7.68 mL | 38.42 mL | 76.84 mL |
| 1 mM | 3.84 mL | 19.21 mL | 38.42 mL |
| 5 mM | 0.77 mL | 3.84 mL | 7.68 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2