Picropodophyllin
目录号: A12195
Picropodophyllin (AXL1717) 是首个针对性的口服小分子 IGF-1 受体抑制剂,对胰岛素受体无影响。
Discription | Picropodophyllin (AXL1717) is the first targeted oral small-molecule IGF-1 receptor inhibitor with no effect on the insulin receptor. | ||
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目录号 | A12195 |
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分子式 | C22H22O8 |
分子量 | 414.4 |
CAS号 | 477-47-4 |
SMILES | COC1=CC(=CC(=C1OC)OC)[C@H]2[C@H]3[C@H](COC3=O)[C@H](C4=CC5=C(C=C24)OCO5)O |
其他名称 | AXL1717, AX-L1717, AXL 1717 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | Warmed: 79 mg/mL (190.63 mM) | |
Water | Insoluble | ||
Ethanol | Warmed: 1 mg/mL | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 24.13 mL | 120.66 mL | 241.31 mL |
0.5 mM | 4.83 mL | 24.13 mL | 48.26 mL |
1 mM | 2.41 mL | 12.07 mL | 24.13 mL |
5 mM | 0.48 mL | 2.41 mL | 4.83 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2