PKI-587 ( Gedatolisib )

目录号: A11079

PI3K/mTOR inhibitor

PKI-587 ( Gedatolisib )

PKI-587 ( Gedatolisib ) Chemical Structure

CAS NO. 1197160-78-3

PKI-587 is a highly potent PI3K/mTOR kinase inhibitor that inhibits PI3K-α,β,γ, δ isoforms and mTOR with IC50 of 0.4, 6.0, 5.4, 6.0 and 1.6 nM respectively.

库存: 现货

规格 价格 数量
5 mg
¥ 500.00
10 mg
¥ 900.00
50 mg
¥ 3,600.00
100 mg
¥ 6,800.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

PKI-587 is a highly potent PI3K/mTOR kinase inhibitor that inhibits PI3K-α,β,γ, δ isoforms and mTOR with IC50 of 0.4, 6.0, 5.4, 6.0 and 1.6 nM respectively.
Targets
PI3Kα (Cell-free assay) mTOR (Cell-free assay) PI3Kγ (Cell-free assay)
0.4 nM1.6 nM5.4 nM
In vitro DMSO 2 mg/mL (3.24 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 16.24 mL 81.21 mL 162.42 mL
0.5 mM 3.25 mL 16.24 mL 32.48 mL
1 mM 1.62 mL 8.12 mL 16.24 mL
5 mM 0.32 mL 1.62 mL 3.25 mL

*The above data is based on the productmolecular weight 615.7. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A11079
MECHANISM OF ACTION Inhibitor
M. Wt 615.7
Formula C32H41N9O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1197160-78-3
Synonyms PKI587, Gedatolisib
SMILES CN(C)C1CCN(CC1)C(=O)C2=CC=C(C=C2)NC(=O)NC3=CC=C(C=C3)C4=NC(=NC(=N4)N5CCOCC5)N6CCOCC6

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