PKI-587 ( Gedatolisib )

目录号: A11079

PI3K/mTOR 抑制剂

PKI-587 ( Gedatolisib )

PKI-587 ( Gedatolisib ) Chemical Structure

CAS NO. 1197160-78-3

PKI-587 (Gedatolisib)是一种高效的PI3K/mTOR激酶抑制剂,可抑制PI3K-α,β,γ,δ亚型和mTOR,IC50分别为0.4、6.0、5.4、6.0和1.6 nM。

库存: 现货

规格 价格 数量
5 mg
¥ 500.00
10 mg
¥ 900.00
50 mg
¥ 3,600.00
100 mg
¥ 6,800.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

PKI-587 (Gedatolisib)是一种高效的PI3K/mTOR激酶抑制剂,可抑制PI3K-α,β,γ,δ亚型和mTOR,IC50分别为0.4、6.0、5.4、6.0和1.6 nM。
靶点信息
PI3Kα (Cell-free assay) mTOR (Cell-free assay) PI3Kγ (Cell-free assay)
0.4 nM1.6 nM5.4 nM
In vitro DMSO 2 mg/mL (3.24 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 16.24 mL 81.21 mL 162.42 mL
0.5 mM 3.25 mL 16.24 mL 32.48 mL
1 mM 1.62 mL 8.12 mL 16.24 mL
5 mM 0.32 mL 1.62 mL 3.25 mL

*The above data is based on the productmolecular weight 615.7. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A11079
作用机制 Inhibitor (抑制剂)
M. Wt 615.7
Formula C32H41N9O4
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 1197160-78-3
Synonyms PKI587, Gedatolisib
SMILES CN(C)C1CCN(CC1)C(=O)C2=CC=C(C=C2)NC(=O)NC3=CC=C(C=C3)C4=NC(=NC(=N4)N5CCOCC5)N6CCOCC6

产品标签

产品标签

其他人对该产品使用了下列标签:

使用空格分隔标签。使用单引号(')标注词组。

Product Questions

Product Questions

No Questions
Keywords:购买 PKI-587 ( Gedatolisib ) | PKI-587 ( Gedatolisib ) 供应商 | 订购 PKI-587 ( Gedatolisib ) | PKI-587 ( Gedatolisib ) 价格 | PKI-587 ( Gedatolisib ) 生产商 | 订单 PKI-587 ( Gedatolisib ) | PKI-587 ( Gedatolisib ) 代理商 | 购买 1197160-78-3| 1197160-78-3 供应商 | 订购 1197160-78-3 | 1197160-78-3 价格 | 1197160-78-3 生产商 | 订单 1197160-78-3 | 1197160-78-3 代理商|buy PKI-587 ( Gedatolisib ) | PKI-587 ( Gedatolisib ) Supplier | purchase PKI-587 ( Gedatolisib ) | PKI-587 ( Gedatolisib ) cost | PKI-587 ( Gedatolisib ) manufacturer | order PKI-587 ( Gedatolisib ) | PKI-587 ( Gedatolisib ) distributor | buy 1197160-78-3| 1197160-78-3 Supplier | purchase 1197160-78-3 | 1197160-78-3 cost | 1197160-78-3 manufacturer | order 1197160-78-3 | 1197160-78-3 distributor
Rewards