(R)-Elagolix

Name: (R)-Elagolix
SKU: A21184

目录号: A21184

GnRHR antagonist

(R)-Elagolix Chemical Structure

CAS NO. 834153-87-6

Elagolix is a highly potent, selective, orally-active, short-duration, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (KD = 54 pM).

库存：现货

规格	价格	数量
2 mg	￥ 540.00
5 mg	￥ 1,080.00
10 mg	￥ 2,100.00
50 mg	￥ 6,180.00

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生物活性

Elagolix is a highly potent, selective, orally-active, short-duration, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (KD = 54 pM).

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	15.83 mL	79.17 mL	158.33 mL
0.5 mM	3.17 mL	15.83 mL	31.67 mL
1 mM	1.58 mL	7.92 mL	15.83 mL
5 mM	0.32 mL	1.58 mL	3.17 mL

*The above data is based on the productmolecular weight 631.59. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A21184
作用机制	Antagonist (拮抗剂)
M. Wt	631.59
Formula	C32H30F5N3O5
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	834153-87-6
Synonyms	NBI-56418, NBI56418, NBI 56418
SMILES	FC1=C(C2=C(C)N(CC3=C(C(F)(F)F)C=CC=C3F)C(N(C[C@](C4=CC=CC=C4)([H])NCCCC(O)=O)C2=O)=O)C=CC=C1OC