Raxatrigine (GSK1014802)

目录号: A13020

Sodium channel blocker

Raxatrigine (GSK1014802)

Raxatrigine (GSK1014802) Chemical Structure

CAS NO. 934240-30-9

Raxatrigine (GSK1014802)是一种新型的钠通道阻滞剂,是一种有效的抗惊厥药物。在大鼠中,GSK1014802(20-80 mg/kg p.o.)以剂量依赖的方式减轻了苯环利定(PCP)诱导的逆向学习障碍,这表明GSK1014802在治疗精神分裂症的认知潜力方面具有潜力。 GSK2还是人MAO-B的有效抑制剂,pIC50值为7.96,但不抑制人MAO-A。

库存: 现货

规格 价格 数量
5 mg
¥ 1,600.00
25 mg
¥ 3,200.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

Raxatrigine (GSK1014802)是一种新型的钠通道阻滞剂,是一种有效的抗惊厥药物。在大鼠中,GSK1014802(20-80 mg/kg p.o.)以剂量依赖的方式减轻了苯环利定(PCP)诱导的逆向学习障碍,这表明GSK1014802在治疗精神分裂症的认知潜力方面具有潜力。 GSK2还是人MAO-B的有效抑制剂,pIC50值为7.96,但不抑制人MAO-A。
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 31.81 mL 159.06 mL 318.12 mL
0.5 mM 6.36 mL 31.81 mL 63.62 mL
1 mM 3.18 mL 15.91 mL 31.81 mL
5 mM 0.64 mL 3.18 mL 6.36 mL

*The above data is based on the productmolecular weight 314.35. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A13020
作用机制 Blocker (阻断剂)
M. Wt 314.35
Formula C18H19FN2O2
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 934240-30-9
Synonyms GSK1014802, GSK-1014802, GSK 1014802
SMILES FC1=CC=CC=C1COC2=CC=C([C@@](N3)([H])CC[C@@]3([H])C(O)=N)C=C2

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