Regadenoson
目录号: A12541
A2A adenosine 激动剂
Regadenoson 是一种选择性的 A2A 腺苷受体 激动剂,相比于 A1、A2B 和 A3 受体,在结合和功能研究中表现出较高的选择性。Regadenoson 还被发现是一种强效的全激动剂,能够引起冠状动脉扩张,这一反应在 A2A 受体 储备中具有很大的潜力。
Discription | Regadenoson was selective agonist for the A2A adenosine receptor versus the A1, A2B, and A3 receptors in binding and functional studies. Regadenoson was also found to be a full and potent agonist to cause coronary vasodilation, a response that has a very large A2A receptor reserve? |
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目录号 | A12541 |
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分子式 | C15H18N8O5 |
分子量 | 390.35 |
CAS号 | 313348-27-5 |
SMILES | C/N=C(O)/C(C=N1)=CN1C2=NC(N)=C(N=CN3[C@@]4([H])[C@@](O)([H])[C@@](O)([H])[C@@](O4)([H])CO)C3=N2 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 49 mg/mL (125.53 mM) | |
Water | Insoluble | ||
Ethanol | 49 mg/mL | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 25.62 mL | 128.09 mL | 256.18 mL |
0.5 mM | 5.12 mL | 25.62 mL | 51.24 mL |
1 mM | 2.56 mL | 12.81 mL | 25.62 mL |
5 mM | 0.51 mL | 2.56 mL | 5.12 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2