Ritanserin
目录号: A21976
5-HT2 receptor 拮抗剂
Ritanserin(R 55667)是一种高效、相对选择性、口服活性、长效的5-HT2受体拮抗剂,其IC50为0.9 nM,对组胺H1、多巴胺D2、肾上腺素能α1、肾上腺素能α2受体的活性较低。
Discription | Ritanserin (R 55667) is a highly potent, relatively selective, orally active, long acting antagonist of 5-HT2 receptor, with an IC50 of 0.9 nM, less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors. | |||||
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Cell Research |
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目录号 | A21976 |
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分子式 | C27H25F2N3OS |
分子量 | 477.57 |
CAS号 | 87051-43-2 |
SMILES | CC1=C(C(N(C=CS2)C2=N1)=O)CCN(CC/3)CCC3=C(C4=CC=C(F)C=C4)\C5=CC=C(F)C=C5 |
其他名称 | R 55667, R55667, R-55667 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2