RPR-260243
目录号: A20977
HERG activator
RPR-260243 是一种新型的 HERG 激活剂;能够修正被多非利多抑制的 HERG 电流(IC50 = 58 nM);对 HERG 电流幅度影响较小,且对稳态激活参数或通道失活过程没有显著影响。
Discription | RPR-260243 is a novel activator of HERG; modifies HERG currents inhibited by dofetilide (IC50 = 58 nM); little effect on HERG current amplitude and no significant effects on steady-state activation parameters or on channel inactivation processes. | |||||
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Cell Research |
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目录号 | A20977 |
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分子式 | C28H25F3N2O4 |
分子量 | 510.5 |
CAS号 | 668463-35-2 |
SMILES | O=C([C@H]1CN(CC#CC2=CC(F)=CC(F)=C2F)CC[C@H]1CCC(C3=CC=NC4=CC=C(OC)C=C34)=O)O |
其他名称 | RPR260243, RPR 260243 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2