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RS 17053 HCl

RS 17053 HCl

Name: RS 17053 HCl
SKU: A16885

目录号: A16885

α1A 拮抗剂

RS 17053 HCl Chemical Structure

CAS NO. 169505-93-5

RS 17053 HCl是α1A受体拮抗剂，对α1A受体具有很高的亲和力（pKi和pA2估计为9.1-9.9），选择性比α1B和α1D亚型高30-100倍（pKi和pA2估计为7.7- 7.8）。

库存：现货

规格	价格	数量
5 mg	￥ 600.00
10 mg	￥ 1,000.00
50 mg	￥ 3,800.00
100 mg	￥ 7,000.00

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生物活性

RS 17053 HCl是α1A受体拮抗剂，对α1A受体具有很高的亲和力（pKi和pA2估计为9.1-9.9），选择性比α1B和α1D亚型高30-100倍（pKi和pA2估计为7.7- 7.8）。

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	22.25 mL	111.25 mL	222.51 mL
0.5 mM	4.45 mL	22.25 mL	44.5 mL
1 mM	2.23 mL	11.13 mL	22.25 mL
5 mM	0.45 mL	2.23 mL	4.45 mL

*The above data is based on the productmolecular weight 449.42. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A16885
作用机制	Antagonist (拮抗剂)
M. Wt	449.42
Formula	C24H29N2O2Cl?HCl
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	169505-93-5
Synonyms	RS-17053, RS17053
SMILES	Cl.CC(C)(CC1=CNC2=CC=C(Cl)C=C12)NCCOC1=C(OCC2CC2)C=CC=C1