RTS-V5
目录号: A20099
HDAC/proteasome 抑制剂
RTS-V5 是一种双重 HDAC/蛋白酶体抑制剂,其 IC50 分别为 HDAC1 6.9 μM、HDAC2 18 μM、HDAC3 15 μM、HDAC6 0.27 μM、HDAC8 0.53 μM。
Discription | RTS-V5 is a dual HDAC/proteasome inhibitor with IC50s of 6.9, 18, 15, 0.27, 0.53 μM for HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, respectively. | |||||
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Cell Research |
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目录号 | A20099 |
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分子式 | C27H35N5O6 |
分子量 | 525.6 |
CAS号 | 2285346-31-6 |
SMILES | O=C(NO)C1=CC=C(C(N[C@@H](CC(NCC(C)(C)C)=O)C(N[C@@H](C)C(NCC2=CC=CC=C2)=O)=O)=O)C=C1 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2