Rupatadine Fumarate

目录号: A12356

PAFR inhibitor/H1 receptor inhibitor

Rupatadine Fumarate Chemical Structure

CAS NO. 182349-12-8

Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 and 102 nM, respectively.

库存: 现货

规格 价格 数量
5 mg
¥ 600.00
10 mg
¥ 1,000.00
25 mg
¥ 2,000.00
50 mg
¥ 3,500.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 and 102 nM, respectively.
Targets
Histamine H1 receptor PAFR
102 nM(Ki)550 nM(Ki)
In vitro (25°C) DMSO 9 mg/mL (16.91 mM)
Water <1 mg/mL (<1 mM)
Ethanol 13 mg/mL (24.43 mM)
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.8 mL 93.98 mL 187.96 mL
0.5 mM 3.76 mL 18.8 mL 37.59 mL
1 mM 1.88 mL 9.4 mL 18.8 mL
5 mM 0.38 mL 1.88 mL 3.76 mL

*The above data is based on the productmolecular weight 532.03. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A12356
MECHANISM OF ACTION Inhibitor
M. Wt 532.03
Formula C26H26ClN3.C4H4O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 182349-12-8
Synonyms N/A
SMILES CC1=CC(=CN=C1)CN2CCC(=C3C4=C(CCC5=C3N=CC=C5)C=C(C=C4)Cl)CC2.C(=C/C(=O)O)\C(=O)O

产品标签

产品标签

其他人对该产品使用了下列标签:

使用空格分隔标签。使用单引号(')标注词组。

Product Questions

Product Questions

No Questions
Keywords:购买 Rupatadine Fumarate | Rupatadine Fumarate 供应商 | 订购 Rupatadine Fumarate | Rupatadine Fumarate 价格 | Rupatadine Fumarate 生产商 | 订单 Rupatadine Fumarate | Rupatadine Fumarate 代理商 | 购买 182349-12-8| 182349-12-8 供应商 | 订购 182349-12-8 | 182349-12-8 价格 | 182349-12-8 生产商 | 订单 182349-12-8 | 182349-12-8 代理商|buy Rupatadine Fumarate | Rupatadine Fumarate Supplier | purchase Rupatadine Fumarate | Rupatadine Fumarate cost | Rupatadine Fumarate manufacturer | order Rupatadine Fumarate | Rupatadine Fumarate distributor | buy 182349-12-8| 182349-12-8 Supplier | purchase 182349-12-8 | 182349-12-8 cost | 182349-12-8 manufacturer | order 182349-12-8 | 182349-12-8 distributor
Rewards