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Saxagliptin (BMS-477118)


DPP-4 抑制剂

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产品目录号: A11109


产品名 目录号 价格 数量
Saxagliptin 10mg A11109-10
¥ 900.00
Saxagliptin 25mg A11109-25
¥ 1,500.00
Saxagliptin 50mg A11109-50
¥ 2,400.00
Saxagliptin 100mg A11109-100
¥ 3,500.00
Saxagliptin (BMS-477118) 10mM * 1mL in DMSO A11109-10mM-D
¥ 910.00



Saxagliptin (BMS-477118) is a new dipeptidyl peptidase-4 (DPP-4) inhibitor with IC50 of 50 nM.

Saxagliptin (BMS-477118)




顾客使用 Adooq 产品发表的高质量科研文献
Adooq 顾客使用 Saxagliptin (BMS-477118) 发表的文献 (2)
  • Chintan N. Koyani, .et al. Saxagliptin but Not Sitagliptin Inhibits CaMKII and PKC via DPP9 Inhibition in Cardiomyocytes, Front Physiol, 2018, 9: 1622 PMID: 30487758
  • Koyani CN, .et al. Dipeptidyl peptidase-4 independent cardiac dysfunction links saxagliptin to heart failure, Biochem Pharmacol, 2016, Dec 1;145:64-80 PMID: 28859968

Chemical Information

目录号 A11109
Mechanism of action Inhibitor
分子量 315.4
化学分子式 C18H25N3O2
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 361442-04-8
Synonyms BMS-477118,Onglyza
SMILES code C1[C@@H]2C[C@@H]2N([C@@H]1C#N)C(=O)[C@H](C34CC5CC(C3)CC(C5)(C4)O)N
化学名称 (1S,3S,5S)-2-[(2S)-2-amino-2-(3-hydroxy-1-adamantyl)acetyl]-2-azabicyclo[3.1.0]hexane-3-carbonitrile


Saxagliptin (BMS-477118) is a new dipeptidyl peptidase-4 (DPP-4) inhibitor with IC50 of 50 nM.
26 nM


Solubility (25°C) * In vitro DMSO 63 mg/mL (199.74 mM)
Water 63 mg/mL (199.74 mM)
Ethanol 24 mg/mL (76.09 mM)
In vivo Saline 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.


Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 31.71 mL 158.53 mL 317.06mL
0.5 mM 6.34 mL 31.71 mL 63.41 mL
1 mM 3.17 mL 15.85 mL 31.71 mL
5 mM 0.63 mL 3.17 mL 6.34 mL

*The above data is based on the productmolecular weight 315.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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