|p38α (Cell-free assay)||p38β (Cell-free assay)|
|50 nM||100 nM|
|In vitro (25°C)||DMSO||66 mg/mL (199.19 mM)|
|Water||<1 mg/mL (<1 mM)|
|Ethanol||12 mg/mL (36.21 mM)|
|In vivo||1% DMSO/30% polyethylene glycol/1% Tween 80||30 mg/mL|
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|0.1 mM||30.18 mL||150.92 mL||301.84 mL|
|0.5 mM||6.04 mL||30.18 mL||60.37 mL|
|1 mM||3.02 mL||15.09 mL||30.18 mL|
|5 mM||0.6 mL||3.02 mL||6.04 mL|
*The above data is based on the productmolecular weight 331.3 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
|MECHANISM OF ACTION||Inhibitor|
|Storage||at -20°C 3 years Powder|
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