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SB 334867

促销

OX1 receptor 拮抗剂

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产品目录号: A12786

库存状态:中国现货中国现货

产品名 目录号 价格 数量
SB 334867 5mg A12786-5
¥ 400.00
SB 334867 10mg A12786-10
¥ 750.00
SB 334867 25mg A12786-25
¥ 1,500.00
SB 334867 50mg A12786-50
¥ 2,500.00

产品仅用于研究,不针对患者销售,望谅解.

产品简介

SB 334867 is a selective non-peptide orexin OX1 receptor antagonist. pKb values are 7.2 and < 5 for inhibition of intracellular Ca2+ release in CHO cells expressing human OX1 and OX2 receptors respectively. Blocks orexin-A induced grooming and feeding following systemic administration in vivo.

SB 334867

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顾客使用 Adooq 产品发表的高质量科研文献
Adooq 顾客使用 SB 334867 发表的文献 (1)
  • Tony Ngo, .et al. Orphan receptor ligand discovery by pickpocketing pharmacological neighbors, Nat Chem Biol, 2017, Feb; 13(2): 235每242 PMID: 27992882

Chemical Information

目录号 A12786
Mechanism of action Antagonist
分子量 319.32
化学分子式 C17H13N5O2
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 249889-64-3
Synonyms SB334867,SB-334867
SMILES code CC1=NC2=C(O1)C=C(C=C2)NC(=O)NC3=C4C(=NC=C3)C=CC=N4
化学名称 N-(2-Methyl-6-benzoxazolyl)-N'-1,5-n?aphthyridin-4-yl urea

生物活性

Description
SB 334867 is a selective non-peptide orexin OX1 receptor antagonist. pKb values are 7.2 and < 5 for inhibition of intracellular Ca2+ release in CHO cells expressing human OX1 and OX2 receptors respectively. Blocks orexin-A induced grooming and feeding following systemic administration in vivo.

制备储备液

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 31.32 mL 156.58 mL 313.17mL
0.5 mM 6.26 mL 31.32 mL 62.63 mL
1 mM 3.13 mL 15.66 mL 31.32 mL
5 mM 0.63 mL 3.13 mL 6.26 mL

*The above data is based on the productmolecular weight 319.32. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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