SB-705498
目录号: A11143
TRPV1 拮抗剂
SB-705498 是一种强效、选择性且口服生物利用度高的 TRPV1 拮抗剂。
| Discription | SB-705498 is a potent, selective and orally bioavailable TRPV1 antagonist. | ||
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| Targets |
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| 目录号 | A11143 |
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| 分子式 | C17H16BrF3N4O |
| 分子量 | 428 |
| CAS号 | 501951-42-4 |
| SMILES | C1CN(C[C@@H]1NC(=O)NC2=CC=CC=C2Br)C3=NC=C(C=C3)C(F)(F)F |
| 其他名称 | SB705498 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
| In vitro | DMSO | 78 mg/mL (181.71 mM) | |
| Water | Insoluble | ||
| Ethanol | 18 mg/mL (41.93 mM) | ||
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 23.36 mL | 116.82 mL | 233.64 mL |
| 0.5 mM | 4.67 mL | 23.36 mL | 46.73 mL |
| 1 mM | 2.34 mL | 11.68 mL | 23.36 mL |
| 5 mM | 0.47 mL | 2.34 mL | 4.67 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2