SCH58261

Name: SCH58261
SKU: A15886

目录号: A15886

A2A adenosine receptor 拮抗剂

SCH58261 Chemical Structure

CAS NO. 160098-96-4

SCH58261是一种有效的选择性A2a腺苷受体拮抗剂，对大鼠A2a和牛A2a的Ki分别为2.3 nM和2 nM。

库存：现货

规格	价格	数量
5 mg	￥ 750.00
10 mg	￥ 1,400.00
25 mg	￥ 2,800.00

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生物活性

SCH58261是一种有效的选择性A2a腺苷受体拮抗剂，对大鼠A2a和牛A2a的Ki分别为2.3 nM和2 nM。

靶点信息

bovine A2a	rat A2a
2.0 nM(Ki)	2.3 nM(Ki)

溶解度 *

In vitro (25°C)	DMSO	61 mg/mL (176.63 mM)
	Water	Insoluble
	Ethanol	Insoluble
In vivo	4% DMSO40% PEG 300+4% Tween 80++ddH2O	1 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	28.96 mL	144.78 mL	289.55 mL
0.5 mM	5.79 mL	28.96 mL	57.91 mL
1 mM	2.9 mL	14.48 mL	28.96 mL
5 mM	0.58 mL	2.9 mL	5.79 mL

*The above data is based on the productmolecular weight 345.36. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A15886
作用机制	Antagonist (拮抗剂)
M. Wt	345.36
Formula	C18H15N7O
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	160098-96-4
Synonyms	SCH-58261, SCH 58261
SMILES	NC1=NC(N(CCC2=CC=CC=C2)N=C3)=C3C4=NC(C5=CC=CO5)=NN14