SEL120-34A HCl
目录号: A21485
CDK8 抑制剂
SEL120-34A HCl 是一种有效的、选择性的、可口服的、ATP竞争性的 CDK8 抑制剂,对 CDK8/CycC 和 CDK19/CycC 的 IC50 分别为 4.4 nM 和 10.4 nM,具有抗肿瘤活性。
Discription | SEL120-34A HCl is a potent, selective, orally available, ATP-competitive CDK8 inhibitor, with IC50s of 4.4 nM and 10.4 nM for CDK8/CycC and CDK19/CycC, respectively, with antitumor activity. | ||
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目录号 | A21485 |
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分子式 | C15H18Br2N4.HCl |
分子量 | 450.6 |
CAS号 | 1609452-30-3 |
SMILES | CC1=C2C3=C(CCCN3C(=N2)N4CCNCC4)C(=C1Br)Br.Cl |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2