SGI 1027

目录号: A14120

DNMT 抑制剂

SGI 1027

SGI 1027 Chemical Structure

CAS NO. 1020149-73-8

SGI 1027是DNMT抑制剂,对DNMT1,DNMT3A和DNMT3B的IC50分别为6、8、7.5 uM。

库存: 现货

规格 价格 数量
10 mg
¥ 900.00
25 mg
¥ 1,800.00
50 mg
¥ 3,100.00
10mM * 1mL in DMSO
¥ 1,100.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

SGI 1027是DNMT抑制剂,对DNMT1,DNMT3A和DNMT3B的IC50分别为6、8、7.5 uM。
靶点信息
DNMT1 (Cell-free assay) DNMT3B (Cell-free assay) DNMT3A (Cell-free assay)
6 μM7.5 μM8 μM
In vitro (25°C) DMSO 85 mg/mL (184.17 mM)
Water Insoluble
Ethanol Insoluble
In vivo 2% DMSO+30% PEG 300+2% Tween 80+ddH2O 1 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.67 mL 108.34 mL 216.68 mL
0.5 mM 4.33 mL 21.67 mL 43.34 mL
1 mM 2.17 mL 10.83 mL 21.67 mL
5 mM 0.43 mL 2.17 mL 4.33 mL

*The above data is based on the productmolecular weight 461.52. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A14120
作用机制 Inhibitor (抑制剂)
M. Wt 461.52
Formula C27H23N7O
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 1020149-73-8
Synonyms SGI-1027, SGI1027
SMILES CC1=CC(=NC(=N1)N)NC2=CC=C(C=C2)NC(=O)C3=CC=C(C=C3)NC4=CC=NC5=CC=CC=C54

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