SHR1653

Name: SHR1653
SKU: A18575

目录号: A18575

Oxytocin receptor antagonist

SHR1653 Chemical Structure

CAS NO. 2231770-73-1

SHR1653 is a highly potent, selective and brain penetrated oxytocin receptor (OTR) antagonist, with an IC50 of 15 nM for hOTR.

库存：现货

规格	价格	数量
5 mg	￥ 3,500.00
10 mg	￥ 6,500.00
50 mg	￥ 20,000.00

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生物活性

SHR1653 is a highly potent, selective and brain penetrated oxytocin receptor (OTR) antagonist, with an IC50 of 15 nM for hOTR.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	23.26 mL	116.31 mL	232.62 mL
0.5 mM	4.65 mL	23.26 mL	46.52 mL
1 mM	2.33 mL	11.63 mL	23.26 mL
5 mM	0.47 mL	2.33 mL	4.65 mL

*The above data is based on the productmolecular weight 429.88. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A18575
作用机制	Antagonist (拮抗剂)
M. Wt	429.88
Formula	C21H21ClFN5O2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	2231770-73-1
Synonyms	SHR 1653, SHR-1653
SMILES	COC1=CC=C(N2C(N3C[C@@]4(C5=CC=C(F)C=C5Cl)C[C@@]4([H])C3)=NN=C2COC)C=N1