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DDP-4 抑制剂

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产品目录号: A14377


产品名 目录号 价格 数量
Sitagliptin 25mg A14377-25
¥ 1,200.00
Sitagliptin 50mg A14377-50
¥ 2,000.00
Sitagliptin 100mg A14377-100
¥ 3,200.00
Sitagliptin 10mM * 1mL in DMSO A14377-10mM-D
¥ 790.00



Sitagliptin is an oral antihyperglycemic (anti-diabetic drug) of the dipeptidyl peptidase-4 (DPP-4) inhibitor class.





顾客使用 Adooq 产品发表的高质量科研文献
Adooq 顾客使用 Sitagliptin 发表的文献 (2)
  • Hae Jin Kim, .et al. Potentiation of endothelium-dependent vasorelaxation of mesenteric arteries from spontaneously hypertensive rats by gemigliptin, a dipeptidyl peptidase-4 inhibitor class of anti-diabetic drug, Korean J Physiol Pharmacol, 2018, Nov; 22(6): 713每719 PMID: 30402032
  • Chintan N. Koyani, .et al. Saxagliptin but Not Sitagliptin Inhibits CaMKII and PKC via DPP9 Inhibition in Cardiomyocytes, Front Physiol, 2018, 9: 1622 PMID: 30487758

Chemical Information

目录号 A14377
Mechanism of action Inhibitor
分子量 407.31
化学分子式 C16H15F6N5O
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 486460-32-6
Synonyms MK-0431, MK 0431, MK0431
SMILES code C1CN2C(=NN=C2C(F)(F)F)CN1C(=O)C[C@@H](CC3=CC(=C(C=C3F)F)F)N
化学名称 (R)-3-amino-1-(3-(trifluoromethyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)-4-(2,4,5-trifluorophenyl)butan-1-one Phosphate Monohydrate


Sitagliptin is an oral antihyperglycemic (anti-diabetic drug) of the dipeptidyl peptidase-4 (DPP-4) inhibitor class.


Solubility (25°C) * In vitro DMSO 100 mg/mL (191.08 mM)
Water 41 mg/mL (78.34 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo Saline 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.


Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.55 mL 122.76 mL 245.51mL
0.5 mM 4.91 mL 24.55 mL 49.1 mL
1 mM 2.46 mL 12.28 mL 24.55 mL
5 mM 0.49 mL 2.46 mL 4.91 mL

*The above data is based on the productmolecular weight 407.31. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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