SR-4835
目录号: A22337
dual 抑制剂 of CDK12/CDK13
SR-4835 是一种强效、高度选择性且与ATP竞争的 CDK12/CDK13 双重抑制剂(CDK12:IC50=99 nM,Kd=98 nM;CDK13:Kd=4.9 nM)。
Discription | SR-4835 is a potent, highly selective and ATP competitive dual inhibitor of CDK12/CDK13 (CDK12: IC50=99 nM, Kd=98 nM; CDK13: Kd=4.9 nM). |
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目录号 | A22337 |
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分子式 | C21H20Cl2N10O |
分子量 | 499.36 |
CAS号 | 2387704-62-1 |
SMILES | CN1N=CC(N2C3=NC(N4CCOCC4)=NC(NCC5=NC6=C(N5)C=C(Cl)C(Cl)=C6)=C3N=C2)=C1 |
其他名称 | SR4835,SR 4835 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2