SRX3207
目录号: A22305
Syk/PI3K 抑制剂
SRX3207 是一种口服活性的首创类双重 Syk/PI3K 抑制剂,其 IC50 值分别针对 Syk 和 PI3Kα 为 10.7 nM 和 861 nM。SRX3207 能够缓解肿瘤免疫抑制。
Discription | SRX3207 is an orally active and first-in-class dual Syk/PI3K inhibitor, with IC50 values of 10.7 nM and 861 nM for Syk and PI3Kα, respectively. SRX3207 relieves tumor immunosuppression. |
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目录号 | A22305 |
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分子式 | C29H29N7O3S |
分子量 | 555.65 |
CAS号 | 2254693-15-5 |
SMILES | O=C1C2=C(C(C3=CC=C(NC4=NC=CC(N5N=C(C)C(CN6CCC6)=C5)=N4)C=C3)=CS2)OC(N7CCOCC7)=C1 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2