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Sulfatinib

Sulfatinib

Name: Sulfatinib
SKU: A21915

目录号: A21915

tyrosine kinase inhibitor

Sulfatinib Chemical Structure

CAS NO. 1308672-74-3

Sulfatinib (HMPL-012) is a potent and highly selective tyrosine kinase inhibitor against VEGFR1/2/3, FGFR1 and CSF1R with IC50s of in a range of 1 to 24 nM.

库存：现货

规格	价格	数量
1 mg	￥ 450.00
5 mg	￥ 1,350.00
10 mg	￥ 2,300.00
50 mg	￥ 6,900.00

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产品仅用于科学研究，不针对患者销售，望谅解.

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生物活性

Sulfatinib (HMPL-012) is a potent and highly selective tyrosine kinase inhibitor against VEGFR1/2/3, FGFR1 and CSF1R with IC50s of in a range of 1 to 24 nM.

溶解度 *

In vitro	DMSO	92 mg/mL (191.43 mM)
	Water	<1 mg/mL
	Ethanol	<1 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	20.81 mL	104.04 mL	208.08 mL
0.5 mM	4.16 mL	20.81 mL	41.62 mL
1 mM	2.08 mL	10.4 mL	20.81 mL
5 mM	0.42 mL	2.08 mL	4.16 mL

*The above data is based on the productmolecular weight 480.58. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A21915
作用机制	Inhibitor (抑制剂)
M. Wt	480.58
Formula	C24H28N6O3S
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1308672-74-3
Synonyms	HMPL-012, HMPL012, HMPL 012
SMILES	O=S(CC1=CC=CC(NC2=NC=CC(OC3=CC4=C(NC(C)=C4)C=C3)=N2)=C1)(NCCN(C)C)=O