T-3775440 hydrochloride
目录号: A18340
LSD1 抑制剂
T-3775440(盐酸盐)是一种不可逆的赖氨酸特异性组蛋白去甲基化酶(LSD1)抑制剂,其IC50值为2.1 nM。
Discription | T-3775440 (hydrochloride) is an irreversible lysine-specific histone demethylase (LSD1) inhibitor with an IC50 value of 2.1 nM. |
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目录号 | A18340 |
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分子式 | C18H23ClN4O |
分子量 | 346.85 |
CAS号 | 1422535-52-1 |
SMILES | O=C(C1=CN(C)N=C1)NC2=CC=C([C@H]3[C@H](NCC4CC4)C3)C=C2.[H]Cl |
其他名称 | T-3775440 HCl; T 3775440 HCl; T3775440 HCl; |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 66 mg/mL (190.28 mM) | |
Water | 21 mg/mL (60.54 mM) | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 28.83 mL | 144.15 mL | 288.31 mL |
0.5 mM | 5.77 mL | 28.83 mL | 57.66 mL |
1 mM | 2.88 mL | 14.42 mL | 28.83 mL |
5 mM | 0.58 mL | 2.88 mL | 5.77 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2