Talnetant
目录号: A15254
NK3 receptor 拮抗剂
Talnetant 是一种强效且选择性的 NK3 受体拮抗剂(ki=1.4 nM, hNK-3-CHO);对 hNK-3 与 hNK-2 受体具有 100 倍的选择性,且在高达 100 uM 的浓度下对 hNK-1 无亲和力。
Discription | Talnetant is a potent and selective NK3 receptor antagonist(ki=1.4 nM, hNK-3-CHO); 100-fold selective for the hNK-3 versus hNK-2 receptor, with no affinity for the hNK-1 at concentrations up to 100 uM. | |||||
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Cell Research |
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目录号 | A15254 |
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分子式 | C25H22N2O2 |
分子量 | 382.45 |
CAS号 | 174636-32-9 |
SMILES | CCC(C1=CC=CC=C1)NC(=O)C2=C(C(=NC3=CC=CC=C32)C4=CC=CC=C4)O |
其他名称 | SB-223412, SB223412, SB 223412 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2