Taranabant
目录号: A11578
CB1 receptor inverse 激动剂
Taranabant 是一种高效且选择性的大麻素1(CB1)受体反向激动剂,能够抑制多种激动剂的结合和功能活性,其对人类CB1R的结合Ki值为0.13 nM。
Discription | Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist that inhibits the binding and functional activity of various agonists, with a binding Ki of 0.13 nM for the human CB1R in vitro. | |||||
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Cell Research |
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目录号 | A11578 |
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分子式 | C27H25ClF3N3O2 |
分子量 | 515.95 |
CAS号 | 701977-09-5 |
SMILES | ClC1=CC=C(C[C@@H](C2=CC=CC(C#N)=C2)[C@@H](NC(C(C)(OC3=CC=C(C=N3)C(F)(F)F)C)=O)C)C=C1 |
其他名称 | MK-0364 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2