Trusted by 10,000+ Scientists since 2006
微信关注
申请试用装

Tedalinab

CB2 receptor 激动剂

0 Customer Reviews
产品目录号: A14189

库存状态:中国现货中国现货

产品名 目录号 价格 数量
Tedalinab 5mg A14189-5
¥ 2,200.00
Tedalinab 10mg A14189-10
¥ 5,000.00
Tedalinab 25mg A14189-25
¥ 9,000.00

产品仅用于研究,不针对患者销售,望谅解.

产品简介

Tedalinab (GRC-10693) is a drug developed for the treatment of osteoarthritis and neuropathic pain, which acts as a potent and selective cannabinoid CB2 receptor agonist. It has a very high selectivity of 4700x for CB2 over the related CB1 receptor, has good oral bioavailability and has shown promising safety results and effective analgesic and antiinflammatory actions in early clinical trials.

Tedalinab

双击上述图片即可查看完整大小

缩小
放大

更多视图

顾客使用 Adooq 产品发表的高质量科研文献

Chemical Information

目录号 A14189
Mechanism of action Agonist
分子量 345.4
化学分子式 C19H21F2N3O
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 916591-01-0
Synonyms GRC-10693
SMILES code CC(C)(C)NC(=O)C1=NN(C2=C1[C@H]3CC[C@@H]2C3)C4=C(C=C(C=C4)F)F
化学名称 (1r,7s)-3-(2,4-difluorophenyl)-n-(2-methyl-2-propanyl)-3,4-diazatricyclo[5.2.1.02,6]deca-2(6),4-diene-5-carboxamide

生物活性

Description
Tedalinab (GRC-10693) is a drug developed for the treatment of osteoarthritis and neuropathic pain, which acts as a potent and selective cannabinoid CB2 receptor agonist. It has a very high selectivity of 4700x for CB2 over the related CB1 receptor, has good oral bioavailability and has shown promising safety results and effective analgesic and antiinflammatory actions in early clinical trials.

制备储备液

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 28.95 mL 144.76 mL 289.52mL
0.5 mM 5.79 mL 28.95 mL 57.9 mL
1 mM 2.9 mL 14.48 mL 28.95 mL
5 mM 0.58 mL 2.9 mL 5.79 mL

*The above data is based on the productmolecular weight 345.4. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Ordering online

To place an order online, simply browse to the product you are interested in and click on the 'Add to Cart' button. To complete this process, you will need to confirm the size and quantity of the products that you require.

To complete an order you will need to register using our simple online registration process. We do not share your contact details with any third parties.

When you are ready to check out simply enter your PO number to complete the ordering process. Please ensure that you send us a copy of your PO by fax or email afterwards.  We will then liaise with you or your purchasing department to confirm the order.

Found your products but not ready to order?

Why not use our WishList feature to store lists of products? This convenient feature allows you to manage lists, append notes to products and share lists with co-workers or colleagues.

Ordering offline

You can email or fax us your purchase order and we will place the order for you. You can also phone us to place the order.  Our contact details are:

We require the following information to process your order:
  • The catalog number for each product. 
  • Your email address or fax number. 
  • Your name and telephone number. 
  • Shipping address and billing address.
  • Purchase order numbers.

产品标签

使用空格分隔标签。使用单引号(')标注词组。


Keywords:购买 Tedalinab | Tedalinab 供应商 | 订购 Tedalinab | Tedalinab 价格 | Tedalinab 生产商 | 订单 Tedalinab | Tedalinab 代理商 | 购买 916591-01-0| 916591-01-0 供应商 | 订购 916591-01-0 | 916591-01-0 价格 | 916591-01-0 生产商 | 订单 916591-01-0 | 916591-01-0 代理商|buy Tedalinab | Tedalinab Supplier | purchase Tedalinab | Tedalinab cost | Tedalinab manufacturer | order Tedalinab | Tedalinab distributor | buy 916591-01-0| 916591-01-0 Supplier | purchase 916591-01-0 | 916591-01-0 cost | 916591-01-0 manufacturer | order 916591-01-0 | 916591-01-0 distributor