Teneligliptin hydrobromide
目录号: A15258
DPP-4 抑制剂
Teneligliptin 是一种新型、高效且持久的二肽基肽酶-4抑制剂;在体外竞争性抑制人类血浆、大鼠血浆和人类重组DPP-4,其IC50值约为1纳摩尔。
| Discription | Teneligliptin is a novel, potent, and long-lasting dipeptidyl peptidase-4 inhibitor; competitively inhibited human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50 values of approximately 1 nM. | ||
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| 目录号 | A15258 |
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| 分子式 | C44H65Br5N12O2S2 |
| 分子量 | 1257.72 |
| CAS号 | 906093-29-6 |
| SMILES | CC1=NN(C(=C1)N2CCN(CC2)C3CC(NC3)C(=O)N4CCSC4)C5=CC=CC=C5.CC1=NN(C(=C1)N2CCN(CC2)C3CC(NC3)C(=O)N4CCSC4)C5=CC=CC=C5.Br.Br.Br.Br.Br |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
| In vitro | DMSO | 85 mg/mL (135.16 mM) | |
| Water | 85 mg/mL (135.16 mM) | ||
| Ethanol | 14 mg/mL | ||
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 7.95 mL | 39.75 mL | 79.51 mL |
| 0.5 mM | 1.59 mL | 7.95 mL | 15.9 mL |
| 1 mM | 0.8 mL | 3.98 mL | 7.95 mL |
| 5 mM | 0.16 mL | 0.8 mL | 1.59 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2